BDBM50063489 CHEMBL3398457
SMILES Cc1oc(nc1CCOc1cccc(CC[C@H]2CN(C[C@@H]2C(O)=O)C(=O)Oc2ccccc2)c1)-c1ccccc1
InChI Key InChIKey=PWZFOKWHYLVOCW-LSYYVWMOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50063489
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to PPARalpha (unknown origin) using fluorescein-tagged dual PPARalpha/gamma activator by homogeneous fluorescence polarization bindi...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Binding affinity to PPARgamma (unknown origin) using fluorescein-tagged dual PPARalpha/gamma activator by homogeneous fluorescence polarization bindi...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataEC50: 1.17E+3nMAssay Description:Agonist activity at GAL4 tagged human PPARgamma ligand binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Agonist activity at GAL4 tagged human PPARalpha ligand binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair