BDBM50078818 1-[4-(3-Ethyl-10-methoxy-8-methyl-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-piperidin-1-yl]-2-(1-oxy-pyridin-4-yl)-ethanone::CHEMBL57728
SMILES CCc1cnc2C(C3CCN(CC3)C(=O)Cc3cc[n+]([O-])cc3)c3c(CCc2c1)cc(C)cc3OC
InChI Key InChIKey=NUMVJPFFYAFXGT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50078818
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair