BDBM50079627 CHEMBL3414768
SMILES NC(=O)c1cccc(NC(=O)C2=C(CCC2)C(O)=O)c1
InChI Key InChIKey=FDQXEDMRIBACLZ-UHFFFAOYSA-N
Data 7 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50079627
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of hexahistidine-tagged human recombinant ARTD7 catalytic domain (459 to 656 amino acids) expressed in Escherichia coli BL21(DE3) assessed...More data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Inhibition of hexahistidine-tagged full length human recombinant ARTD1 expressed in Escherichia coli BL21(DE3) assessed as Inhibition of ADP-ribosylt...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of hexahistidine-tagged human recombinant ARTD8 catalytic domain (1611 to 1801 amino acids) expressed in Escherichia coli BL21(DE3) assess...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of hexahistidine-tagged human recombinant ARTD7 catalytic domain (459 to 656 amino acids) expressed in Escherichia coli BL21(DE3) assessed...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of hexahistidine-tagged full length human recombinant ARTD10 expressed in Escherichia coli BL21(DE3) assessed as Inhibition of ADP-ribosyl...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of hexahistidine-tagged full length human recombinant ARTD10 expressed in Escherichia coli BL21(DE3) assessed as Inhibition of ADP-ribosyl...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of hexahistidine-tagged full length human recombinant ARTD1 expressed in Escherichia coli BL21(DE3) assessed as Inhibition of ADP-ribosylt...More data for this Ligand-Target Pair