BDBM50080291 (5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-pyridin-4-ylmethyl-amine::CHEMBL81863
SMILES Cc1[nH]c2nc(nc(NCc3ccncc3)c2c1C)-c1ccccc1
InChI Key InChIKey=GSAIXPLBVQLLNN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50080291
Affinity DataKi: 132nMAssay Description:Inhibitory activity against binding of the [3H]-DPCPX to human A1 receptor (hA1) radioligands using competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 811nMAssay Description:Inhibitory activity against binding of the [3H]-CGS-21,680 to human A2a receptor (hA2a) radioligands using competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 222nMAssay Description:Inhibitory activity against binding of [3H]-DPCPX to human A1 receptor (hA1) using competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 262nMAssay Description:Inhibitory activity against membranes from HEK293 cells stably expressing the human A2a receptor (hA2a)More data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibitory activity against binding of the [3H]-CGS-21,680 to human A2a receptor (hA2a) radioligands using competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibitory activity against binding of [3H]-DPCPX to human A1 receptor (hA1) using competition binding assayMore data for this Ligand-Target Pair