BDBM50096220 CHEMBL3593635
SMILES [H][C@]12CC[C@]([H])(CC(=C1)c1cnc(NCc3ccc4CCOc4c3)c(c1)C(=O)NCc1ccc(OC)c(Cl)c1)N(C2)C(C)=O
InChI Key InChIKey=ZJRKLCDOMLGCGK-COBDYTDYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50096220
Affinity DataIC50: 5.90nMAssay Description:Displacement of [125I]human ghrelin from rat ghrelin receptor expressed in CHO cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inverse agonist activity rat ghrelin receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Asubio Pharma
Curated by ChEMBL
Asubio Pharma
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Displacement of [125I]human ghrelin from human ghrelin receptor expressed in CHO cell membranes incubated for 30 mins by scintillation counting metho...More data for this Ligand-Target Pair