BDBM50097410 CHEMBL3586450

SMILES CN1CCN(CC1)c1cncc(c1)-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1

InChI Key InChIKey=CHKLDGFTXXDTQV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50097410   

TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50097410(CHEMBL3586450)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human METAP2 using Met-Pro-Arg-pNa substrate by para-nitroanilide chromophore release detection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed