BDBM50107018 CHEMBL108070::N-(4-Methyl-benzoyl)-N'-(2-thiophen-2-yl-ethyl)-guanidine

SMILES Cc1ccc(cc1)C(=O)NC(N)=NCCc1cccs1

InChI Key InChIKey=QBQQLAJXKVUTGB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50107018   

TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cenes Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50107018(CHEMBL108070 | N-(4-Methyl-benzoyl)-N'-(2-thiophen...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Cenes Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50107018(CHEMBL108070 | N-(4-Methyl-benzoyl)-N'-(2-thiophen...)
Affinity DataIC50:  4.95E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed