BDBM50112174 CHEMBL3608430

SMILES [H][C@@]12CN(C[C@]1([H])CN(C2)c1nc(Nc2ccc(cc2)N2CCN(C)CC2)c2ncn(C(C)C)c2n1)C(=O)C=C

InChI Key InChIKey=CBZIPGPDJXMUAK-OYRHEFFESA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50112174   

TargetEpidermal growth factor receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50112174(CHEMBL3608430)
Affinity DataIC50:  181nMAssay Description:Inhibition of wild type EGFR in human A549 cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed