BDBM50113369 CHEMBL286421::N-{4-[(R)-1-(3-Cyclopentyloxy-4-methoxy-phenyl)-2-pyridin-4-yl-ethyl]-phenyl}-2,3,4,5,6-pentafluoro-benzenesulfonamide

SMILES COc1ccc(cc1OC1CCCC1)[C@H](Cc1ccncc1)c1ccc(NS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1

InChI Key InChIKey=BTUWFPWOMKRTNQ-HSZRJFAPSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50113369   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50113369(CHEMBL286421 | N-{4-[(R)-1-(3-Cyclopentyloxy-4-met...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed