BDBM50129169 9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::9-bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline::CHEMBL294265

SMILES COc1cc(Br)cc-2c1OCc1c-2ccc2NC(C)(C)C=C(C)c12

InChI Key InChIKey=MZIFJAQJEZFKDE-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50129169   

TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129169(9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6...)
Affinity DataKi:  476nMAssay Description:Binding affinity at human progesterone receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129169(9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6...)
Affinity DataKi:  479nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129169(9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6...)
Affinity DataEC50:  43nMAssay Description:Antagonistic activity at human progesterone receptor in CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed