BDBM50137133 4,6-Bis-benzoylamino-isophthalic acid::CHEMBL156717::NS3763

SMILES OC(=O)c1cc(C(O)=O)c(NC(=O)c2ccccc2)cc1NC(=O)c1ccccc1

InChI Key InChIKey=UUDYZUDTQPLDDP-UHFFFAOYSA-N

Data  6 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50137133   

TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch

Curated by PDSP Ki Database
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed