BDBM50154947 CHEMBL3774757
SMILES Cn1cc(cn1)-c1ccc(Cc2n[nH]c3ccc(cc23)-c2nccn2C)cc1
InChI Key InChIKey=BGVLCUOYRCTJCU-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50154947
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of CDK8 (unknown origin) expressed in 7dF3 clone of human HEK293 cells preincubated for 2 hrs followed by addition of beta-estradiol by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Displacement of dye-labeled ATP competitive probe from recombinant human CDK8/Cyclin C incubated for 20 mins by Alexa647 probe-based FRET assayMore data for this Ligand-Target Pair