BDBM50158030 4-[6-Chloro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine::CHEMBL360234

SMILES Nc1ccc(cc1)S(=O)(=O)n1cc(C2=CCNCC2)c2ccc(Cl)cc12

InChI Key InChIKey=NWRMZTXFSRHJFJ-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50158030   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50158030(4-[6-Chloro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-in...)
Affinity DataKi:  3nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cells using [3H]-LSDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50158030(4-[6-Chloro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-in...)
Affinity DataIC50:  11.2nMAssay Description:Inhibitory concentration against 5-HT stimulated cAMP production in HeLa cells stably transfected with human 5-HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed