BDBM50159451 CHEMBL216992::Des-AA1,2,5,12,13-[D-Trp8]SRIF

SMILES C[C@@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](N)CSSC[C@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)C(O)=O

InChI Key InChIKey=ANCUAJMQRRZZNC-JFMJRBFYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50159451   

TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159451(CHEMBL216992 | Des-AA1,2,5,12,13-[D-Trp8]SRIF)
Affinity DataIC50:  13nMAssay Description:Inhibition of 125I-[Leu8,D-Trp22,Tyr25]SRIF-28 binding to human somatostatin receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159451(CHEMBL216992 | Des-AA1,2,5,12,13-[D-Trp8]SRIF)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of 125I-[Leu8,D-Trp22,Tyr25]SRIF-28 binding to human somatostatin receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159451(CHEMBL216992 | Des-AA1,2,5,12,13-[D-Trp8]SRIF)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of 125I-[Leu8,D-Trp22,Tyr25]SRIF-28 binding to human somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159451(CHEMBL216992 | Des-AA1,2,5,12,13-[D-Trp8]SRIF)
Affinity DataIC50:  15nMAssay Description:Inhibition of 125I-[Leu8,D-Trp22,Tyr25]SRIF-28 binding to human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159451(CHEMBL216992 | Des-AA1,2,5,12,13-[D-Trp8]SRIF)
Affinity DataIC50:  39nMAssay Description:Inhibition of 125I-[Leu8,D-Trp22,Tyr25]SRIF-28 binding to human somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed