BDBM50170197 CHEMBL367359::N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-fluoro-benzamide

SMILES CN(C)c1nc(N[C@@H]2CC[C@@H](CC2)NC(=O)c2ccccc2F)nc2ccccc12

InChI Key InChIKey=AGEXNHZEGLFEDD-IYBDPMFKSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50170197   

TargetMelanin-concentrating hormone receptor 1(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50170197(CHEMBL367359 | N-[4-(4-Dimethylamino-quinazolin-2-...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against human CA-MCH-R1 (Melanin-concentrating hormone receptor 1) by using [125I](Phe13,Tyr19)MCH as radioligand expressed in HE...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed