BDBM50174860 4-(3-Bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-1-(2-pyridin-4-yl-acetyl)-piperazine-2-carboxylic acid cyclopropylmethyl-amide::CHEMBL425032

SMILES Clc1ccc2C(N3CCN(C(C3)C(=O)NCC3CC3)C(=O)Cc3ccncc3)c3ncc(Br)cc3CCc2c1

InChI Key InChIKey=KGSICNXNFOBMJP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50174860   

LigandPNGBDBM50174860(4-(3-Bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cycl...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed