BDBM50186367 CHEMBL379959::c(his-D-phe-arg-trp-Ahp)

SMILES NC(=N)NCCC[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](Cc2cnc[nH]2)NC(=O)CCCCCCNC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O

InChI Key InChIKey=YQBUXOUSHPXETO-LDLFXXLYSA-N

Data  1 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50186367   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataKi:  244nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataEC50:  67nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataEC50:  15.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed