BDBM50186367 CHEMBL379959::c(his-D-phe-arg-trp-Ahp)
SMILES NC(=N)NCCC[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](Cc2cnc[nH]2)NC(=O)CCCCCCNC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O
InChI Key InChIKey=YQBUXOUSHPXETO-LDLFXXLYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50186367
Affinity DataKi: 244nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 15.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair