BDBM50198913 CHEMBL1179089
SMILES C(COC(c1ccccc1)c1ccccc1)Cc1c[nH]cn1
InChI Key InChIKey=LJIRQKCQUPMGIY-UHFFFAOYSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50198913
Affinity DataKi: 17nMAssay Description:Displacement of [125I]iodoproxyfan from human H3 receptor expressed in HEK293 cell membranes after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Antagonist activity at H3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity at human H4 receptor expressed in CHO cells co-expressing Galphai2 assessed as inhibition of imetit-induced GTPgamma[35S] binding...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...More data for this Ligand-Target Pair