BDBM50216663 (R)-N-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-phenyl-2-(phenylsulfonamido)propanamide::CHEMBL393019

SMILES CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](Cc2ccccc2)NS(=O)(=O)c2ccccc2)C1=O)c1ccccc1

InChI Key InChIKey=NMNCSFDNUCUWFV-UHSQPCAPSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50216663   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50216663((R)-N-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Blockade of human Nav1.7 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed