BDBM50216673 CHEMBL246195::tert-butyl (R)-1-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-ylamino)-1-oxo-4-phenylbutan-2-ylcarbamate
SMILES CN1c2ccccc2C(=N[C@@H](NC(=O)[C@@H](CCc2ccccc2)NC(=O)OC(C)(C)C)C1=O)c1ccccc1
InChI Key InChIKey=GASQNNOBMSQSOK-SQHAQQRYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50216673
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:Blockade of human Nav1.7 by FRET assayMore data for this Ligand-Target Pair