BDBM50224207 2-(2-fluorophenylamino)-5-isopropylthiazol-4(5H)-one::CHEMBL392452::CHEMBL393908::CHEMBL396617
SMILES CC(C)c1sc(Nc2ccccc2F)nc1O
InChI Key InChIKey=XHOHMOHZBDGVBQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50224207
Affinity DataKi: 7nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human 11betaHSD1 in CHO cells assessed as conversion of cortisone to cortisolMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of human 11betaHSD1 in CHO cells assessed as conversion of cortisone to cortisolMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human 11betaHSD1 in CHO cells assessed as conversion of cortisone to cortisolMore data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of human 11betaHSD1 in presence of 3% HSA by cell based assayMore data for this Ligand-Target Pair