BDBM50236548 CHEMBL4097535
SMILES Oc1ccc(cc1)-c1cnc2[nH]cc(C(=O)Nc3cccc(O)c3)c2c1
InChI Key InChIKey=CMLCCTPKLYKIJA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50236548
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity to the human androgen receptor (hAR) in CV-1 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assayMore data for this Ligand-Target Pair