BDBM50253845 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide::CHEMBL517116

SMILES CCc1c(nn(c1-c1ccc(s1)C#CCC(C)C)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1

InChI Key InChIKey=IXEWYTLXTLCWOK-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50253845   

TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50253845(1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-...)
Affinity DataIC50:  5.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50253845(1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-...)
Affinity DataEC50:  23nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50253845(1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-...)
Affinity DataIC50:  1.21E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed