BDBM50256396 CHEMBL4079208
SMILES Cc1[nH]c(c2CCCC(=O)c12)-c1cc(ccc1Oc1ccc(F)cc1F)S(C)(=O)=O
InChI Key InChIKey=RFRKNJZNTDDXFX-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50256396
Affinity DataKi: 460nMAssay Description:Binding affinity to His-tagged BRD4 BD1-BD2 (K57 to K550 residues) (unknown origin) after 1 hr by Alexa-647-conjugated probe based TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in human H1299 cells co-expressing HPV16-LCR/E2 after 24 hrs by Bright Glo-luciferase reporter gene ass...More data for this Ligand-Target Pair