BDBM50259240 (5-(1-Benzyl-1H-indazol-3-yl)-1,2,4-oxadiazol-3-yl)methanamine::CHEMBL512079
SMILES NCc1noc(n1)-c1nn(Cc2ccccc2)c2ccccc12
InChI Key InChIKey=VUXLKOATKUTQHW-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50259240
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human Nav1.6 expressed in HEK293 cells assessed as change in membrane potential using MP-red voltage sensitve dyeMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair