BDBM50264534 CHEMBL4075311::US10005735, Table 1.6

SMILES Sc1cccc2ncccc12

InChI Key InChIKey=XAXWWYIMGUQNMY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50264534   

Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM50264534(CHEMBL4075311 | US10005735, Table 1.6)
Affinity DataIC50: >1.00E+5nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM50264534(CHEMBL4075311 | US10005735, Table 1.6)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed