BDBM50293980 (R)-5-Chloro-1-(1-cyclopropylethyl)-3-[(2,6-dichloro-4-methoxyphenyl)(ethyl)amino]pyrazin-2(1H)-one::CHEMBL563618

SMILES CCN(c1nccn([C@H](C)C2CC2)c1=O)c1c(Cl)cc(OC)cc1Cl

InChI Key InChIKey=ACZGTUUOYXZHMJ-LLVKDONJSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50293980   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293980((R)-5-Chloro-1-(1-cyclopropylethyl)-3-[(2,6-dichlo...)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed