BDBM50299249 1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde::CHEMBL583972::US8481586, 3
SMILES O=Cc1c[nH]c2c1ccc1c3ccccc3[nH]c21
InChI Key InChIKey=VWNCOFUKBTYAON-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50299249
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 120nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 510nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 10nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 120nMAssay Description:Inhibition of human Pim1 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 510nMAssay Description:Inhibition of human GST fused Pim2 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 120nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 510nMAssay Description:Inhibition of human Pim2 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent
Affinity DataIC50: 10nMAssay Description:Inhibition of human Pim3 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Centre National De La Recherche Scientifique
US Patent
Centre National De La Recherche Scientifique
US Patent