BDBM50301030 CHEMBL567679::N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-methyl-2-(4-(trifluoromethyl)pyridin-2-ylamino)propanamide
SMILES C[C@H](NC(=O)C(C)(C)Nc1cc(ccn1)C(F)(F)F)[C@@H](Cc1ccc(Cl)cc1)c1cccc(c1)C#N
InChI Key InChIKey=YYHJKDYUEKFPTH-GAJHUEQPSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50301030
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair
Affinity DataIC50: 353nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair