BDBM50304273 2-((2S,4S)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)-4-hydroxypyrrolidin-2-yl)acetic acid::CHEMBL593039
SMILES [#6]-c1ccsc1\[#6](=[#6]/[#6]-[#6]-[#7]-1-[#6]-[#6@@H](-[#8])-[#6]-[#6@H]-1-[#6]-[#6](-[#8])=O)-c1sccc1-[#6]
InChI Key InChIKey=LJBQPELFQMHCCO-HOTGVXAUSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50304273
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Institute Of Microbiology
Curated by ChEMBL
Institute Of Microbiology
Curated by ChEMBL
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of GAT1 in mouse D8 cells assessed as [3H]GABA transport by liquid scintillation countingMore data for this Ligand-Target Pair