BDBM50318545 Ac-ARAEVH-NH2::CHEMBL1086454

SMILES CC(C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(N)=O

InChI Key InChIKey=AFTMQAFHRKDEPI-CMQAMBHRSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50318545   

TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318545(Ac-ARAEVH-NH2 | CHEMBL1086454)
Affinity DataKi:  90nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318545(Ac-ARAEVH-NH2 | CHEMBL1086454)
Affinity DataIC50:  400nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed