BDBM50331432 CHEMBL1289527::N-{3-[(1,1-Dioxo-1H-1lambda*6*-benzo[d]isothiazol-3-yl)-phenyl-amino]-propyl}-nicotinamide

SMILES O=C(NCCCN(C1=NS(=O)(=O)c2ccccc12)c1ccccc1)c1cccnc1

InChI Key InChIKey=KHQIQPQMMQPOOI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50331432   

TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331432(CHEMBL1289527 | N-{3-[(1,1-Dioxo-1H-1lambda*6*-ben...)
Affinity DataIC50:  2.75E+3nMAssay Description:Inhibition of human voltage-gated potassium channel Kv1.3 expressed in CGE22 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed