BDBM50334721 3-Amino-N-(3-(naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)propanamide HCl::CHEMBL1642867

SMILES NCCC(=O)Nc1ccc2c(n[nH]c2c1)S(=O)(=O)c1cccc2ccccc12

InChI Key InChIKey=LLZGCYHPURCHJM-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50334721   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334721(3-Amino-N-(3-(naphthalen-1-ylsulfonyl)-1H-indazol-...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-LSD from cloned human 5-HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50334721(3-Amino-N-(3-(naphthalen-1-ylsulfonyl)-1H-indazol-...)
Affinity DataIC50:  456nMAssay Description:Antagonist activity at cloned human 5-HT6 receptor expressed in human HeLa cells assessed as inhibition of 5HT-induced cyclic AMP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed