BDBM50336937 3-[(4-methoxyphenyl)phenylmethyl]indole::CHEMBL1672540

SMILES COc1ccc(cc1)C(c1c[nH]c2ccccc12)c1ccccc1

InChI Key InChIKey=BTEQZWJLBYEBLQ-UHFFFAOYSA-N

Data  4 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50336937   

TargetGlucocorticoid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  50.2nMAssay Description:Displacement of [3H]methyltrienolone from human glucocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  68.9nMAssay Description:Displacement of [3H]methyltrienolone from human androgen receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  86.8nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataKi:  478nMAssay Description:Displacement of [3H]methyltrienolone from human progesterone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataIC50:  3.72E+3nMAssay Description:Antagonist activity at human progesterone receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by GRE-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336937(3-[(4-methoxyphenyl)phenylmethyl]indole | CHEMBL16...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed