BDBM50339765 CHEMBL1689122::rac-2-(4-chloro-2-((2-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
SMILES CC1CN(CCN1Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)c1ccccc1
InChI Key InChIKey=KQVTZYFUHDWJOQ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50339765
Affinity DataIC50: 71nMAssay Description:Antagonist activity against human CRTh2 receptor expressed in CHO cells assessed as inhibition of PGD2-mediated Ca2+ fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair