BDBM50347766 CHEMBL1802849

SMILES CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCC1CC1

InChI Key InChIKey=OBKVROGZKBOQSW-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50347766   

TargetDual specificity protein kinase CLK1(Mus musculus)
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  130nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Mus musculus)
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  510nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK3 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  340nMAssay Description:Inhibition of human recombinant GST-tagged DYRK2 using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant Pim1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Universite£? De Rennes 1

Curated by ChEMBL
LigandPNGBDBM50347766(CHEMBL1802849)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed