BDBM50373614 CHEMBL257288

SMILES CC(C)OC(=O)C1C(N(CCCN(C)C(=O)c2ccc(Oc3ccccc3)cc2)C(=O)N=C1C)c1cccc(Cl)c1

InChI Key InChIKey=SMLIUJCIWNKLJV-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50373614   

TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Bristol-Myers Squibb R & D

Curated by ChEMBL
LigandPNGBDBM50373614(CHEMBL257288)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at human alpha1H T-type calcium channel expressed in HEK293 cells by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Bristol-Myers Squibb R & D

Curated by ChEMBL
LigandPNGBDBM50373614(CHEMBL257288)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at human alpha1H T-type calcium channel expressed in HEK293 cells by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Bristol-Myers Squibb R & D

Curated by ChEMBL
LigandPNGBDBM50373614(CHEMBL257288)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at human alpha1H T-type calcium channel expressed in HEK293 cells by patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed