BDBM50383254 CHEMBL2032201

SMILES Cn1cnc2C(N(CCc12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C(F)(F)F

InChI Key InChIKey=ZSTGYKXUKMGRAN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50383254   

TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Amgen

Curated by ChEMBL
LigandPNGBDBM50383254(CHEMBL2032201)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior icilin inductio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed