BDBM50400521 CHEMBL2204933

SMILES Cc1nc(no1)[C@@H]1N[C@H](Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccc(F)cc1

InChI Key InChIKey=RMUNXROCBCEXAA-WIYYLYMNSA-N

Data  1 KI  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50400521   

LigandPNGBDBM50400521(CHEMBL2204933)
Affinity DataKi:  2.21E+3nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400521(CHEMBL2204933)
Affinity DataIC50:  29nMAssay Description:Inhibition of mouse SSTR3 transfected in CHO cells assessed as inhibition of SRIF-induced reduction of cAMP accumulation after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400521(CHEMBL2204933)
Affinity DataIC50:  8.10nMAssay Description:Displacement of [125I]SS-28 from mouse SSTR3 transfected in CHO cells after 60 to 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400521(CHEMBL2204933)
Affinity DataIC50:  58nMAssay Description:Inhibition of human SSTR3 transfected in CHO cells assessed as inhibition of SRIF-induced reduction of cAMP accumulation after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400521(CHEMBL2204933)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [125I]SS-28 from human SSTR3 transfected in CHO cells after 60 to 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed