BDBM50405123 CHEMBL4175898

SMILES COc1ccc(NC2(C(=O)N(C3CCCCC3)C(=O)C2=Cc2ccccc2)c2cccc(Cl)c2)cc1OC

InChI Key InChIKey=SAYBAKTYBZIPAL-MSOSYJBYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50405123   

TargetHistamine H3 receptor(Homo sapiens (Human))
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405123(CHEMBL4175898)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human H3R expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405123(CHEMBL4175898)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human H3R expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed