BDBM50406882 CHEMBL4166554

SMILES OC(=O)c1nc2ccccc2nc1Nc1ccccc1O

InChI Key InChIKey=XVRFKJJGGJBRMI-UHFFFAOYSA-N

Data  7 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50406882   

TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Pig)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50:  740nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed