BDBM50409950 CHEMBL2096788

SMILES FC(F)(F)c1cccc(c1)C(=O)NCC(=O)NC[C@H]1CCCN1Cc1ccc(Cl)cc1

InChI Key InChIKey=XAFZUHZKNKPLQG-LJQANCHMSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50409950   

TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50:  570nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50:  570nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed