BDBM50419680 CHEMBL1945039
SMILES COc1ccccc1CNCc1cccc(CCNC[C@H](O)c2ccc(O)c3[nH]c(=O)sc23)c1
InChI Key InChIKey=VKCKAMBPNXKGHL-QFIPXVFZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50419680
Affinity DataIC50: 6.30nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Binding affinity to Alpha-1D adrenoreceptor expressed in HEK cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of radiolabeled iodocyanopindolol from beta1 adrenoceptorMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Binding affinity to dopamine D2 receptor expressed in HEK cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Binding affinity to Alpha-1D adrenoceptor expressed in HEK cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to dopamine D2 receptor expressed in HEK cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.501nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig trachea assessed as reduction in methacholine-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Binding affinity to beta1 adrenoceptor expressed in CHO cells by cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.631nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in H292 cells assessed as increase in cAMP accumulation after 60 mins by spectrophotometryMore data for this Ligand-Target Pair