BDBM50420504 CHEMBL2086507
SMILES Fc1ccc(COC(=O)N2CCN(CC2)S(=O)(=O)c2ccc(NC(=O)C=C)cc2)cc1
InChI Key InChIKey=FHKFISJKLJDQGA-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50420504
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human recombinant TG1 by fluorescent transamidation assayMore data for this Ligand-Target Pair