BDBM50426291 CHEMBL2312681

SMILES N[C@@H](C[C@@H](CCNC(=O)OCc1ccccc1)C(O)=O)C(O)=O

InChI Key InChIKey=FOWLPLJQDVNWOP-NEPJUHHUSA-N

Data  3 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50426291   

TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataKi:  217nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataKi:  3.04E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK2(VCR) receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells by [3H]-D-Asp uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells by [3H]-D-Asp uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50426291(CHEMBL2312681)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of human EAAT2 expressed in HEK293 cells by [3H]-D-Asp uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed