BDBM50426534 CHEMBL2323944

SMILES COC(=O)C(C)(C)c1ccc(cc1)N1CCC(CC1)n1c(NC(C)C)nc2c(C(=O)N(C)C)c(Cl)c(Cl)cc12

InChI Key InChIKey=REMGFZJNRXPOSB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50426534   

TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50426534(CHEMBL2323944)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human recombinant TRPV4 expressed in BacMam virus infected HEK MSRII cells assessed as inhibition of GSK1016790A-induced calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed