BDBM50428551 CHEMBL2337513
SMILES CNC(=O)c1ccc(cn1)[C@]1(O)CCN([C@H]1C)c1ccc(C#N)c(Cl)c1
InChI Key InChIKey=ZZRUBPUOTYXWMT-BUXKBTBVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50428551
Affinity DataIC50: 44nMAssay Description:Inhibition of wild type Androgen receptor (unknown origin) expressed in Freestyle293F cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at wild type Androgen receptor in human LNCaP-hr cells assessed as prostate specific antigen secrection measured after 3 days by enz...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to bicalutamide-resistant Androgen receptor T878A mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Binding affinity to wild-type Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at wild type Androgen receptor (unknown origin) expressed in human Cos-7 cells co-expressing pGL3-MMTV-luc vector assessed as luc...More data for this Ligand-Target Pair