BDBM50451762 CHEMBL2112920
SMILES CCCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)NCC(N)=O
InChI Key InChIKey=VGEQKPIZLOMRBH-SSNHPIBPSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50451762
Affinity DataEC50: 25nMAssay Description:Effective concentration against hMC4R using HEK293 cells was determined by measuring cAMP accumulationMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration of compound was determined against hMC1R through displacement of NDP-MSH radioligand using HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Effective concentration against hMC1R using HEK293 cells was determined by measuring the cAMP accumulationMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Effective concentration against hMC1R using HEK293 cells was determined by measuring the cAMP accumulationMore data for this Ligand-Target Pair