BDBM50458816 CHEMBL4203162
SMILES CC[C@H](C)[C@H](NC(=O)[C@H]1Cc2ccc(O)c(CC=CCCNCCCC[C@H](N)C(=O)N[C@@H](CCCCN)C(=O)N3CCC[C@H]3C(=O)N1)c2)C(=O)N[C@@H](CC(C)C)C(O)=O
InChI Key InChIKey=MUYSUNAYXFRSCD-ZGQNLQJXSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50458816
Affinity DataKi: 305nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human NTS1 receptor expressed in CHOK1 cell membranes after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Agonist activity at Galpha13-Rluc2/Gbeta1/GFP10-Ggamma1 fused human NTS1 expressed in CHO-K1 cell membranes assessed as Galpha13 activation after 5 m...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at GFP10/beta-arrestin2-Rluc2 fused human NTS1 expressed in CHO-K1 cell membranes assessed as beta-arrestin2 recruitment after 20 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at Galphaq-Rluc2/Gbeta1/GFP10-Ggamma1 fused human NTS1 expressed in CHO-K1 cell membranes assessed as Galphaq activation after 5 min...More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at GFP10/beta-arrestin1-Rluc2 fused human NTS1 expressed in CHO-K1 cell membranes assessed as beta-arrestin1 recruitment after 20 mi...More data for this Ligand-Target Pair