BDBM50469250 CHEMBL4281351
SMILES [H][C@@]12C[C@@]3([H])C[C@@](CNc4nc(NCc5ccccc5Br)ncc4C#N)(C1)C[C@@]([H])(C2)[C@H]3N
InChI Key InChIKey=MIWMFPOJJJMAJT-PTRWISQFSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50469250
Affinity DataIC50: 31nMAssay Description:Inhibition of PKCtheta in human Jurkat cells transfected with pGL3-IL2 pro 43 plasmid assessed as suppression of IL-2 production after 14 hrs by fire...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair